A general method for the metal-free, regioselective, remote C–H halogenation of 8-substituted quinolines DR Motati, D Uredi, EB Watkins Chemical Science 9 (7), 1782-1788, 2018 | 122 | 2018 |
Rh-catalyzed, regioselective, C–H bond functionalization: access to quinoline-branched amines and dimers MD Reddy, FR Fronczek, EB Watkins Organic letters 18 (21), 5620-5623, 2016 | 111 | 2016 |
Synthesis of 3-substituted and 3, 4-disubstituted pyrazolin-5-ones JC Jung, EB Watkins, MA Avery Tetrahedron 58 (18), 3639-3646, 2002 | 88 | 2002 |
The epothilones and related analogues-a review of their syntheses and anti-cancer activities EB Watkins, AG Chittiboyina, JC Jung, MA Avery Current pharmaceutical design 11 (13), 1615-1653, 2005 | 69 | 2005 |
Synthesis and cyclization reaction of pyrazolin-5-one derivatives JC Jung, EB Watkins, MA Avery Heterocycles: an international journal for reviews and communications in …, 2005 | 66 | 2005 |
Generation of Oxamic Acid Libraries: Antimalarials and Inhibitors of Plasmodium falciparum Lactate Dehydrogenase S Choi, AB Beeler, A Pradhan, EB Watkins, JM Rimoldi, B Tekwani, ... Journal of combinatorial chemistry 9 (2), 292-300, 2007 | 63 | 2007 |
Palladium-Catalyzed Direct Arylation of C(sp3)–H Bonds of α-Cyano Aliphatic Amides MD Reddy, EB Watkins The Journal of Organic Chemistry 80 (22), 11447-11459, 2015 | 59 | 2015 |
A unified strategy for the synthesis of β-carbolines, γ-carbolines, and other fused azaheteroaromatics under mild, metal-free conditions D Uredi, DR Motati, EB Watkins Organic letters 20 (20), 6336-6339, 2018 | 52 | 2018 |
Palladium-Catalyzed, N-(2-Aminophenyl)acetamide-Assisted Ortho-Arylation of Substituted Benzamides: Application to the Synthesis of Urolithins B, M6, and M7 MD Reddy, AN Blanton, EB Watkins The Journal of Organic Chemistry 82 (10), 5080-5095, 2017 | 46 | 2017 |
Recent developments in the syntheses of the epothilones and related analogues EB Watkins, AG Chittiboyina, MA Avery European journal of organic chemistry 2006 (18), 4071-4084, 2006 | 44 | 2006 |
A simple, tandem approach to the construction of pyridine derivatives under metal-free conditions: a one-step synthesis of the monoterpene natural product,(−)-actinidine D Uredi, DR Motati, EB Watkins Chemical communications 55 (22), 3270-3273, 2019 | 37 | 2019 |
Gram-scale, stereoselective synthesis and biological evaluation of (+)-armillariol C MD Reddy, H Kobori, T Mori, J Wu, H Kawagishi, EB Watkins Journal of natural products 80 (9), 2561-2565, 2017 | 36 | 2017 |
Design, synthesis, and biological evaluation of inhibitors of the NADPH oxidase, Nox4 Q Xu, AA Kulkarni, AM Sajith, D Hussein, D Brown, OF Güner, MD Reddy, ... Bioorganic & medicinal chemistry 26 (5), 989-998, 2018 | 34 | 2018 |
First synthesis of antimalarial Machaeriols A and B AG Chittiboyina, CR Reddy, EB Watkins, MA Avery Tetrahedron letters 45 (8), 1689-1691, 2004 | 33 | 2004 |
Addition of lithioimidazoles to isocyanates followed by Pd-coupling: access to 4-substituted imidazole-2, 5-dicarboxamides AG Chittiboyina, CR Reddy, EB Watkins, MA Avery Tetrahedron letters 45 (9), 1869-1872, 2004 | 26 | 2004 |
1,3-Diaxially Substituted trans-Decalins: Potential Nonsteroidal Human Progesterone Receptor Inhibitors Z Li, EB Watkins, H Liu, AG Chittiboyina, PB Carvalho, MA Avery The Journal of Organic Chemistry 73 (19), 7764-7767, 2008 | 25 | 2008 |
Design, Synthesis and Evaluation of Trisubstituted Thiazoles Targeting Plasmodium Falciparum Cysteine Proteases PM Goud, A Sheri, PV Desai, EB Watkins, B Tekwani, Y Sabnis, J Gut, ... Medicinal Chemistry Research 14, 74-105, 2005 | 24 | 2005 |
Solenopsin A and analogs exhibit ceramide-like biological activity I Karlsson, X Zhou, R Thomas, AT Smith, MY Bonner, P Bakshi, AK Banga, ... Vascular cell 7, 1-11, 2015 | 23 | 2015 |
Efficient synthesis of 4-ethoxycarbonyl pyrazolin-5-one derivatives JC Jung, EB Watkins, MA Avery Synthetic communications 32 (24), 3767-3777, 2002 | 19 | 2002 |
Development and validation of a UPLC method for rapid and simultaneous analysis of proton pump inhibitors RT Addo, K Davis, R Ubale, JS Owen, EB Watkins AAPS PharmSciTech 16, 30-34, 2015 | 14 | 2015 |